Enviar artigo por via de e-mail Synthesis of Phosphoisosteres of Amyloid Dipeptide Components
- Autores: Golovash S.R.1, Ivanov D.E.1, Borodachev A.V.1, Shestov V.I.1, Dmitriev M.E.1, Ragulin V.V.1
-
Afiliações:
- Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
- Edição: Volume 94, Nº 1 (2024)
- Páginas: 98-104
- Seção: Articles
- URL: https://cardiosomatics.ru/0044-460X/article/view/667244
- DOI: https://doi.org/10.31857/S0044460X24010081
- EDN: https://elibrary.ru/HKVRCB
- ID: 667244
Citar
Texto integral
Acesso aberto
Acesso está concedido
Acesso é pago ou somente para assinantes
Resumo
A simple and effective method was proposed for the synthesis of new phosphinic peptides in free form, structural isosteres of the dipeptide components of beta-amyloid (Aβ42), potential inhibitors of zinc-metalloproteinases.
Texto integral
Sobre autores
S. Golovash
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Email: rvalery@dio.ru
Rússia, Chernogolovka
D. Ivanov
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Email: rvalery@dio.ru
Rússia, Chernogolovka
A. Borodachev
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Email: rvalery@dio.ru
ORCID ID: 0000-0002-3458-5129
Rússia, Chernogolovka
V. Shestov
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Email: rvalery@dio.ru
Rússia, Chernogolovka
M. Dmitriev
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Email: rvalery@dio.ru
ORCID ID: 0000-0001-8870-195X
Rússia, Chernogolovka
V. Ragulin
Institute of Physiologically Active Compounds, Federal Research Center of Problems of Chemical Physics and Medicinal Chemistry of the Russian Academy of Sciences
Autor responsável pela correspondência
Email: rvalery@dio.ru
ORCID ID: 0000-0002-3967-1034
Rússia, Chernogolovka
Bibliografia
- Collinsova M., Jiracek J. // Curr. Med. Chem. 2000. Vol. 7. N 6. P. 629. doi: 10.2174/0929867003374831
- Dive V., Georgiadis D., Matziari M., Makaritis A., Beau F., Cuniasse P., Yiotakis A. // Cell. Mol. Life Sci. 2004. Vol. 61. P. 2010. doi: 10.1007/s00018-004-4050-y
- Mucha A. // Molecules. 2012. Vol. 17. P. 13530. doi: 10.3390/molecules171113530
- Georgiadis D., Dive V. // Top. Curr. Chem. 2015. Vol. 360. P. 1. doi: 10.1007/128_2014_571
- Zinc Metalloproteases in Health and Disease // Ed. N.M. Hooper. London: Taylor and Francis, 1996. P. 153.
- Hori M., Nishida K. // Cardiovasc. Res. 2009. Vol. 81. N 3. P. 457. doi: 10.1093/cvr/cvn335
- Whittaker M., Ayscough A. // Celltransmissions. 2001. Vol. 17. N 1. P. 3.
- Pirad B., Matter H. // J. Med. Chem. 2006. Vol. 49. N 1. P. 51. doi: 10.1021/jm050363f
- Dafnis I., Argyri L., Chroni A. // Neuroscience. 2018. Vol. 394. P. 144. doi: 10.1016/j.neuroscience.2018.10.026
- Sun X., Chen W.-D., Wang Y.-D. // Front. Pharmacol. 2015. Vol. 6. P. 1. doi: 10.3389/fphar.2015.00221
- Xiong Z.M., Kitagawa K., Nishiuchi Y., Kimura T., Nakamura T., Inagaki C. // Life Sci. 2009. Vol. 84. P. 132. doi: 10.1016/j.lfs.2008.11.011
- Xiong Z.M., Kitagawa K., Nishiuchi Y., Kimura T., Inagaki C. // Neurosci. Lett. 2007. Vol. 419. N 3. P. 247. doi: 10.1016/j.neulet.2007.04.022
- Musiek E.S., Holtzman D.M. // Neuroscience. 2015. Vol. 18. P. 800. doi: 10.1038/nn.4018
- Dafnis I., Argyri L., Sagnou M., Tzinia A., Tsilibary E.C., Stratikos E., Chroni A. // Sci Rep. 2016. Vol. 6. P. 30654. doi: 10.1038/srep30654
- Argyri L., Dafnis I., Theodossiou T.A., Gantz D., Stratikos E., Chroni A. // J. Biol. Chem. 2014. Vol. 289. P.12931. doi: 10.1074/jbc.M113.538124
- Дмитриев М.Э., Рагулин В.В. // ЖОХ. 2015. Т. 85. Вып. 9. С. 1511; Dmitriev M.E., Ragulin V.V. // Russ. J. Gen. Chem. 2015. Vol. 85. N 9. P. 2091. doi: 10.1134/S1070363215090121
- Dmitriev M.E., Golovash S.R., Borodachev A.V., Ragulin V.V. // J. Org. Chem. 2021. Vol. 86. N 1. P.593. doi: 10.1021/acs.joc.0c02259
- Rozhko L.F., Ragulin V.V. // Amino Acids. 2005. Vol. 29. P.139. doi: 10.1007/s00726-005-0194-9
- Dmitriev M.E., Ragulin V.V. // Tetrahedron Lett. 2010. Vol. 51. N 19. P. 2613. doi: 10.1016/j.tetlet.2010.03.020
- Dmitriev M.E., Ragulin V.V. // Tetrahedron Lett. 2012. Vol. 53. N 13. P. 1634. doi: 10.1016/j.tetlet.2012.01.094
Arquivos suplementares
